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Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

Advanced Drug Delivery Reviews · 1997 · Vol. 23(1-3) · pp. 3–25
Christopher A. LipinskiFranco LombardoBeryl W. DominyPaul J. Feeney
Crystallization and Solubility StudiesAnalytical Chemistry and ChromatographyComputational Drug Discovery MethodsSolubilityDrug discoveryChemistryThermodynamicsPermeability (electromagnetism)Hildebrand solubility parameterPermeationWork (physics)Computational chemistryOrganic chemistry
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