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Structure–activity relationship study of bone morphogenetic protein (BMP) signaling inhibitors

Bioorganic & Medicinal Chemistry Letters · 2008 · Vol. 18(15) · pp. 4388–4392
Gregory D. CunyPaul B. YuJoydev K. LahaXuechao XingJifeng LiuCarol LaiDonna Y. DengChetana SachidanandanKenneth D. BlochRandall T. Peterson
TGF-β signaling in diseasesParathyroid Disorders and TreatmentsHeterotopic Ossification and Related ConditionsChemistryBone morphogenetic proteinPyrimidinePiperazineSMADPhosphorylationIn vivoBone morphogenetic protein 2QuinolineStereochemistry

MeSH terms

AnimalsFemaleMalePiperazinesPyrazolesPyrimidinesStructure-Activity RelationshipMolecular StructureSignal TransductionBone Morphogenetic ProteinsCombinatorial Chemistry TechniquesMiceBone Morphogenetic Protein Receptors

Funding

  • Harvard NeuroDiscovery Center
  • Pulmonary Hypertension Association
  • GlaxoSmithKline
  • National Institutes of Health
Citations
337
FWCI
5.24
field-weighted impact
References
36
Percentile
96%
vs. same field & year
Citations per year
References
Role of AMP-activated protein kinase in mechanism of metformin action
Journal of Clinical Investigation · 2001 · 5,364 citations
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