reviewTop 1% cited

Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins

Trends in Pharmacological Sciences · 1993 · Vol. 14(8) · pp. 303–307

Robert J. Lefkowitz✉(Duke University Hospital)Susanna CotecchiaPhilippe Samama(Howard Hughes Medical Institute)Tommaso Costa(Istituto Superiore di Sanità)

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Receptor Mechanisms and Signaling Neuroscience and Neuropharmacology Research Circadian rhythm and melatoninAllosteric regulationReceptorG protein-coupled receptorG proteinTernary complexCell biologyChemistryBiochemistryBiologyBiophysics

MeSH terms

Amino Acid SequenceAnimalsModels, ChemicalMolecular Sequence DataMutationReceptors, Cell SurfaceStereoisomerismStructure-Activity RelationshipGTP-Binding Proteins

Citations

805

FWCI

12.72

field-weighted impact

References

Percentile

99%

vs. same field & year

Citations per year

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References

A Quantitative Analysis of Beta-Adrenergic Receptor Interactions: Resolution of High and Low Affinity States of the Receptor by Computer Modeling of Ligand Binding Data

Molecular Pharmacology · 1980 · 555 citations

Opiate Receptor Binding of Agonists and Antagonists Affected Differentially by Sodium

Molecular Pharmacology · 1974 · 575 citations

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